Российские ученые усовершенствовали препарат для лечения рака предстательной железы
Российские ученые установили, что пространственная структура молекул бикалутамида изменяется в зависимости от используемого растворителя. Этот препарат, широко применяемый при лечении рака предстательной железы, имеет множество различных конформеров, условно поделенных на две группы: «открытые» и «закрытые». Исследователи из Института химии растворов имени Г.А. Крестова РАН (Иваново) изучили, как характеристики растворителя влияют на соотношение этих форм.
«Осмысление пространственной структуры бикалутамида в разных растворителях позволит снизить побочные эффекты препарата. Это может привести к созданию более эффективных и безопасных противораковых лекарственных форм, что, в свою очередь, улучшит качество жизни пациентов», — сообщил руководитель проекта, доктор физико-математических наук и заведующий лабораторией ЯМР-спектроскопии растворов и флюидов Института химии растворов им. Г.А. Крестова РАН, Илья Ходов.
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Thank you for your sharing. I am worried that I lack creative ideas. It is your article that makes me full of hope. Thank you. But, I have a question, can you help me?
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